From: Pharmacological characterisation of murine α4β1δ GABAA receptors expressed in Xenopus oocytes
EC 50 (μM) (pEC 50 ± SEM) | IC 50 (μM) (pIC 50 ± SEM) | n H (± SEM) | N | |
---|---|---|---|---|
GABA | ||||
α4β1δ | 0.89 (6.05 ± 0.05) | 1.1 ± 0.11 | 6 | |
α4β1 | 2.7 (5.56 ± 0.05) | 0.87 ± 0.079 | 5 | |
Zn 2+ | ||||
α4β1δ | 3.3 (5.48 ± 0.03) | −0.75 ± 0.041 | 6 | |
α4β1a | IC 50A | 6 | ||
0.00013 (9.87 ± 0.22) | ND | |||
IC 50B | ||||
0.056 (7.25 ± 0.13) | -1.1 ± 0.13 | |||
Cu 2+ | ||||
α4β1δ | 0.82 (6.09 ± 0.04) | −1.2 ± 0.13 | 12 | |
SCS | ||||
α4β1δ | 0.0042 (8.37 ± 0.25) | 4 |