Table 1 EC50values for agonist-stimulated Ca i ++ release
| Â | 5-HT2AR | 5-HT2CR | ||
|---|---|---|---|---|
| Â | Serum-starved | Serum-replete | Serum-starved | Serum-replete |
5-HT | 0.8 nM | 53 nM | 0.7 nM | 4.9 nM |
DOI | 3.6 nM | > 24 μM | 5.4 nM | > 100 μM |
MK212 | No response | No response | > 280 nm | > 11 μM |